Copyright (c) 2016 AJC
This work is licensed under a Creative Commons Attribution 4.0 International License.
One Pot Synthesis and Antibacterial Activity of (4Z)-4-Benzylidene-1-methyl-2-styryl-1H-imidazol-5(4H)-one
Corresponding Author(s) : V. Anitha Rani
Asian Journal of Chemistry,
Vol. 28 No. 7 (2016): Vol 28 Issue 7
Abstract
Green synthesis of (4Z)-4-benzylidene-1-methyl-2-styryl-1H-imidazol-5(4H)-one derivatives have been developed in good yields and tested for their antibacterial activities against Escherichia coli, Providencia aeruginosa, Pseudomonas azotogensis and Baccilus subtillis. Some of the synthesized compounds possess good activity against Escherichia coli and Baccilus subtillis compared to standard drug streptomycin.
Keywords
Download Citation
Endnote/Zotero/Mendeley (RIS)BibTeX
- B.R. Shah, J.J. Bhatt, H.H. Patel, N.K. Undavia, P.B. Trivedi and N.C. Desai, Indian J. Chem., 34B, 201 (1995).
- I. Krezel, Farmaco, 53, 342 (1998); doi:10.1016/S0014-827X(98)00031-7.
- H.-T. Nguyen, C. Destrade and J. Malthécte, J. Adv. Mater, 9, 375 (1997); doi:10.1002/adma.19970090503.
- H. Joshi, P. Upadhyay, D. Karia and A.J. Baxi, Eur. J. Med. Chem., 38, 837 (2003); doi:10.1016/S0223-5234(03)00117-X.
- H. Miyachi, H. Kiyota and M. Segawa, Bioorg. Med. Chem. Lett., 8, 1807 (1998); doi:10.1016/S0960-894X(98)00312-6.
- K. Borisch, S. Diele, P. Göring, H. Kresse and C. Tschierske, J. Mater. Chem., 8, 529 (1998); doi:10.1039/a705359b.
- D. Mukerji, S.R. Nautiyal and C.R. Prasad, Indian Drugs, 18, 125 (1981).
- A. Solankee, K. Kapadiya, I. Thakor, J. Patel and S. Lad, Asian J. Chem., 16, 917 (2006).
- N.C. Desai, D. Dave, M.D. Shah and G.D. Vyas, Indian J .Chem., 39B, 277 (2000).
- K.V. Hirpara, S.P. Patel, K.A. Parikh, A.S. Bhimani and H.H. Parekh, J. Sci. Islam Rep. Iran, 15, 135 (2004).
- Aydogan and M. Kutlu, Biologia, 62, 6 (2007); doi:10.2478/s11756-007-0008-5.
- N.C. Desai, A.M. Bhavsar and B.B. Baldaniya, Indian J. Pharm. Sci., 71, 90 (2009); doi:10.4103/0250-474X.51953.
- H.M. Imtiaz, V. Kumar, Indian J. Chem., 31B, 285 (1992).
- B. List, R.A. Lerner and C.F. Barbas, J. Am. Chem. Soc., 122, 2395 (2000); doi:10.1021/ja994280y.
- M. Yamaguchi, N. Yokota and T. Minami, J. Chem. Soc. Chem. Commun., 1088 (1991); doi:10.1039/C39910001088.
- Y.Y. Peng, Q.P. Ding, Z. Li, P.G. Wang and J.-P. Cheng, Tetrahedron Lett., 44, 3871 (2003); doi:10.1016/S0040-4039(03)00692-0.
- G.J. Collee, G.A. Fraser, P.B. Marmion and A. Simmons, Practical Medical Microbiology, Churchill Livingstone: Edinburgh, edn 14, vol. 11, p. 163 (1996).
References
B.R. Shah, J.J. Bhatt, H.H. Patel, N.K. Undavia, P.B. Trivedi and N.C. Desai, Indian J. Chem., 34B, 201 (1995).
I. Krezel, Farmaco, 53, 342 (1998); doi:10.1016/S0014-827X(98)00031-7.
H.-T. Nguyen, C. Destrade and J. Malthécte, J. Adv. Mater, 9, 375 (1997); doi:10.1002/adma.19970090503.
H. Joshi, P. Upadhyay, D. Karia and A.J. Baxi, Eur. J. Med. Chem., 38, 837 (2003); doi:10.1016/S0223-5234(03)00117-X.
H. Miyachi, H. Kiyota and M. Segawa, Bioorg. Med. Chem. Lett., 8, 1807 (1998); doi:10.1016/S0960-894X(98)00312-6.
K. Borisch, S. Diele, P. Göring, H. Kresse and C. Tschierske, J. Mater. Chem., 8, 529 (1998); doi:10.1039/a705359b.
D. Mukerji, S.R. Nautiyal and C.R. Prasad, Indian Drugs, 18, 125 (1981).
A. Solankee, K. Kapadiya, I. Thakor, J. Patel and S. Lad, Asian J. Chem., 16, 917 (2006).
N.C. Desai, D. Dave, M.D. Shah and G.D. Vyas, Indian J .Chem., 39B, 277 (2000).
K.V. Hirpara, S.P. Patel, K.A. Parikh, A.S. Bhimani and H.H. Parekh, J. Sci. Islam Rep. Iran, 15, 135 (2004).
Aydogan and M. Kutlu, Biologia, 62, 6 (2007); doi:10.2478/s11756-007-0008-5.
N.C. Desai, A.M. Bhavsar and B.B. Baldaniya, Indian J. Pharm. Sci., 71, 90 (2009); doi:10.4103/0250-474X.51953.
H.M. Imtiaz, V. Kumar, Indian J. Chem., 31B, 285 (1992).
B. List, R.A. Lerner and C.F. Barbas, J. Am. Chem. Soc., 122, 2395 (2000); doi:10.1021/ja994280y.
M. Yamaguchi, N. Yokota and T. Minami, J. Chem. Soc. Chem. Commun., 1088 (1991); doi:10.1039/C39910001088.
Y.Y. Peng, Q.P. Ding, Z. Li, P.G. Wang and J.-P. Cheng, Tetrahedron Lett., 44, 3871 (2003); doi:10.1016/S0040-4039(03)00692-0.
G.J. Collee, G.A. Fraser, P.B. Marmion and A. Simmons, Practical Medical Microbiology, Churchill Livingstone: Edinburgh, edn 14, vol. 11, p. 163 (1996).