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Vol. 31 No. 1 (2019): Vol 31 Issue 1

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Novel Synthesis of 5-Oxo-2-thioxo-2,5-dihydro-3-thiophenecarboxylate Derivatives in Non-Aqueous Medium

https://doi.org/10.14233/ajchem.2019.21622
Nitin Srivastava
Department of Chemistry, Amity University Uttar Pradesh, Lucknow Campus, Lucknow-226028, India
M. Saxena
Department of Chemistry, Amity University Uttar Pradesh, Lucknow Campus, Lucknow-226028, India

Corresponding Author(s) : Nitin Srivastava

nsrivastava1@lko.amity.edu

Asian Journal of Chemistry, Vol. 31 No. 1 (2019): Vol 31 Issue 1

Abstract

A novel synthetic method of synthesis of 5-oxo-2-thioxo-2,5-dihydro-3-thiophenecarboxylate (rhodanine) derivative is being reported using primary amines and acetylenic ester, carbon disufide and Triton-B in non-aqueous medium.

Keywords

Carbon disulfide Primary amine Acetylenic ester Triton-B
Srivastava, N., & Saxena, M. (2018). Novel Synthesis of 5-Oxo-2-thioxo-2,5-dihydro-3-thiophenecarboxylate Derivatives in Non-Aqueous Medium. Asian Journal of Chemistry, 31(1), 176–180. https://doi.org/10.14233/ajchem.2019.21622
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References
  1. Y. Inamori, Y. Okamoto, Y. Takegawa, H. Tsujibo, Y. Sakagami, Y. Kumeda, M. Shibata and A. Numata, Biosci. Biotechnol. Biochem., 62, 1025 (1998); https://doi.org/10.1271/bbb.62.1025.
  2. J. Miao, C.-J. Zheng, L.-P. Sun, M.-X. Song, L.-L. Xu and H.-R. Piao, Med. Chem. Res., 22, 4125 (2013); https://doi.org/10.1007/s00044-012-0417-z.
  3. P. Mitra and A.S. Mitra, J. Indian Chem. Soc., 61, 77 (1984).
  4. A.A. Khalek, C.R. Ashby Jr., B.A. Patel, T.T. Talele and M.N. Seleem, PLoS One, 11, e0164227 (2016); https://doi.org/10.1371/journal.pone.0164227.
  5. W. Sing, C.L. Lee, S.L. Yeo, S.P. Lim and M.M. Sim, Bioorg. Med. Chem. Lett., 11, 91 (2001); https://doi.org/10.1016/S0960-894X(00)00610-7.
  6. M.G. Orchard, J.C. Neuss, C.M. Galley, A. Carr, D.W. Porter, P. Smith, D.I.C. Scopes, D. Haydon, K. Vousden, C.R. Stubberfield, K. Young and M. Page, Bioorg. Med. Chem. Lett., 14, 3975 (2004); https://doi.org/10.1016/j.bmcl.2004.05.050.
  7. N.S. Cutshall, C. O’ Day and M. Prezhdo, Bioorg. Med. Chem. Lett., 15, 3374 (2005); https://doi.org/10.1016/j.bmcl.2005.05.034.
  8. J.H. Ahn, S.J. Kim, W.S. Park, S.Y. Cho, J.D. Ha, S.S. Kim, S.K. Kang, D.G. Jeong, S.-K. Jung, S.-H. Lee, H.M. Kim, S.K. Park, K.H. Lee, C.W. Lee, S.E. Ryu and J.-K. Choi, Bioorg. Med. Chem. Lett., 16, 2996 (2006); https://doi.org/10.1016/j.bmcl.2006.02.060.
  9. E.B. Grant, D. Guiadeen, E.Z. Baum, B.D. Foleno, D.A. Montenegro, H. Jin, E.A. Nelson, K. Bush and D.J. Hlasta, Bioorg. Med. Chem. Lett., 10, 2179 (2000); https://doi.org/10.1016/S0960-894X(00)00444-3.
  10. N.J. Gaikwad and P. Gautam, Indian J. Heterocycl. Chem., 12, 181 (2002).
  11. S.K. Shukla, S.P. Singh, L.P. Awasthi and D.D. Mukherjee, Indian J. Pharm. Sci., 44, 153 (1982).
  12. B.B. Lohray, V. Bhushan, P.B. Rao, G.R. Madhavan, N. Murali, K.N. Rao, G.R. Madhavan, N. Murali, K.N. Rao, K. Anantha Reddy, B.M. Rajesh, P. Ganpathy Reddy, R. Chakrabarti and R. Rajagopalan, Bioorg. Med. Chem. Lett., 7, 785 (1997); https://doi.org/10.1016/S0960-894X(97)00118-2.
  13. S.P. Singh, S.S. Parmar, K. Raman and V.I. Stenberg, Chem. Rev., 81, 175 (1981); https://doi.org/10.1021/cr00042a003.
  14. C.L. Lee and M.M. Sim, Tetrahedron Lett., 41, 5729 (2000); https://doi.org/10.1016/S0040-4039(00)00866-2.
  15. F.C. Brown, Chem. Rev., 61, 463 (1961); https://doi.org/10.1021/cr60213a002.
  16. W.-D. Rudorf and R. Schwarz, Hetrocycles, 24, 3459 (1986); https://doi.org/10.3987/R-1986-12-3459.
  17. S. Gabillet, D. Lecercle, O. Loreau, M. Carboni, S. Dezard, J. Gomis and M. Taran, Org. Lett., 9, 3925 (2007); https://doi.org/10.1021/ol701563e.
  18. A. Alizadeh, F. Movahedi, H. Masrouri and L.-G. Zhu, Synthesis, 3431 (2006); https://doi.org/10.1055/s-2006-950234.
  19. A. Alizadeh, F. Movahedi and A.A. Esmaili, Tetrahedron Lett., 47, 4469 (2006); https://doi.org/10.1016/j.tetlet.2006.04.040.
  20. J. Liu, Y. Zhou, Y. Wu, X. Li and A.S.C. Chan, Tetrahedron Asymm., 19, 832 (2008); https://doi.org/10.1016/j.tetasy.2008.03.015.
  21. D. Kaminskyy, A. Kryshchyshyn and R. Lesyk, Expert Opin. Drug Discov., 12, 1233 (2017); https://doi.org/10.1080/17460441.2017.1388370.
  22. S.S. Alneyadi, Heterocycles, 96, 803 (2018); https://doi.org/10.3987/REV-17-878.
  23. T. Tomasic and L.P. Masiè, Expert Opin. Drug Discov., 7, 549 (2012); https://doi.org/10.1517/17460441.2012.688743.
  24. T. Tomasic and L.P. Masiè, Curr. Med. Chem., 16, 1596 (2009); https://doi.org/10.2174/092986709788186200.
  25. A. Alizadeh, S. Rostamnia, N. Zohreh and R. Hosseinpour, Tetrahedron Lett., 50, 1533 (2009); https://doi.org/10.1016/j.tetlet.2008.12.107.
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