Synthesis and Antimicrobial Activity of Novel Benzisothiazolin-3-one Acetamide Derivatives

Jun Hu; Minjie Yu; Peng Yu; Yanhua Xu

doi:10.14233/ajchem.2014.17594

Issue

Vol. 26 No. 22 (2014): Vol 26 Issue 22

Issue Published : November 6, 2014

This work is licensed under a Creative Commons Attribution 4.0 International License.

Synthesis and Antimicrobial Activity of Novel Benzisothiazolin-3-one Acetamide Derivatives

https://doi.org/10.14233/ajchem.2014.17594

Jun Hu

College of Biology and the Environment, Nanjing Forestry University, Nanjing, P.R. China ; College of Environment, Nanjing University of Technology, Nanjing, P.R. China

Minjie Yu

College of Environment, Nanjing University of Technology, Nanjing, P.R. China

Peng Yu

College of Environment, Nanjing University of Technology, Nanjing, P.R. China

Yanhua Xu

College of Environment, Nanjing University of Technology, Nanjing, P.R. China

Corresponding Author(s) : Yanhua Xu

yhxu2008@163.com

Asian Journal of Chemistry, Vol. 26 No. 22 (2014): Vol 26 Issue 22
Article Published : November 6, 2014

Abstract

A series of novel 2-(3-oxobenzo[d]isothiazol-2(3H)-yl)-N-substituted phenylacetamide (4a-4e) have been synthesized from benzo [d]isothiazol-3(2H)-one (BIT) and substituted aniline. These benzisothiazolin-3-one acetamide derivatives (4a-4e) were identified by IR, ¹H NMR and elemental analyses. Their antimicrobial activities were also evaluated.

Keywords

Synthesis Antimicrobial activity Benzisothiazolin-3-one Acetamide

Hu, J., Yu, M., Yu, P., & Xu, Y. (2014). Synthesis and Antimicrobial Activity of Novel Benzisothiazolin-3-one Acetamide Derivatives. Asian Journal of Chemistry, 26(22), 7680–7682. https://doi.org/10.14233/ajchem.2014.17594

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References

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References

M. Shimizu, T. Shimazaki, T. Yoshida, W. Ando and T. Konakahara, Tetrahedron, 68, 3932 (2012); doi:10.1016/j.tet.2012.03.094.

R.M. Novick, M.L. Nelson, K.M. Unice, J.J. Keenan and D.J. Paustenbach, Food Chem. Toxicol., 56, 60 (2013); doi:10.1016/j.fct.2013.02.006.

H. Herbst, Material Having Antibacterial and Antifungal Properties, US Patent 12/083,054 (2006).

R. Dams, S. Paulussen, D. Vangeneugden and D. Sheel, Method for Depositing a Biocidal Coating on a Substrate, US Patent 13/806,663 (2011).

V.R. Naik and H.B. Naik, Asian J. Chem., 12, 1358 (2000).

V.M. Barot and S.D. Desai, Asian J. Chem., 21, 6091 (2009).

M.K. Ahirwar and S.P. Shrivastava, Asian J. Chem., 22, 7493 (2010).

H. Khalid, Aziz-ur-Rehman, M.A. Abbasi, A. Malik, S. Rasool, K. Nafeesa, I. Ahmad and S. Afzal, J. Saudi Chem. Soc., doi:10.1016/j.jscs.2013.05.001.

M.R. Gannarapu, S.B. Vasamsetti, N. Punna, N.K. Royya, S.R. Pamulaparthy, J.B. Nanubolu, S. Kotamraju and N. Banda, Eur. J. Med. Chem., 143, 75 (2014).

G.G. Berest, O.Y. Voskoboynik, S.I. Kovalenko, O.M. Antypenko, I.S. Nosulenko, A.M. Katsev and O.S. Shandrovskaya, Eur. J. Med. Chem., 46, 6066 (2011); doi:10.1016/j.ejmech.2011.10.022.

M.K. Ibrahim, A.A. Abd-Elrahman, R.R.A. Ayyad, K. El-Adl, A.M. Mansour and I.H. Eissa, Bull. Fac. Pharm. Cairo Univ., 51, 101 (2013); doi:10.1016/j.bfopcu.2012.11.003.

C. Orek, P. Koparir and M. Koparir, Spectrochim. Acta A, 97, 923 (2012); doi:10.1016/j.saa.2012.07.082.

E. Hernández-Núñez, H. Tlahuext, R. Moo-Puc, H. Torres-Gómez, R. Reyes-Martínez, R. Cedillo-Rivera, C. Nava-Zuazo and G. Navarrete-Vazquez, Eur. J. Med. Chem., 44, 2975 (2009); doi:10.1016/j.ejmech.2009.01.005.

M.N. Indu, A.A.M. Hatha, C. Abirosh, U. Harsha and G. Vivekanandan, Braz. J. Microbiol., 37, 153 (2006); doi:10.1590/S1517-83822006000200011.

Issue

Vol. 26 No. 22 (2014): Vol 26 Issue 22

Synthesis and Antimicrobial Activity of Novel Benzisothiazolin-3-one Acetamide Derivatives

Corresponding Author(s) : Yanhua Xu

Abstract

Keywords

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