Biginelli Reaction-Carboxylic Acids as Catalysts

Sadia Noreen; Saima Perveen; Muhammad Naeem Khan; Areesha Nazeer; Misbahul Ain Khan; Munawar Ali Munawar; Rabia Babar; Farah Suhail; Muhammad Azad; Alice M.R. Bernardino; Maurício  S. Dos Santos

doi:10.14233/ajchem.2013.14094

Issue

Vol. 25 No. 9 (2013): Vol 25 Issue 9

Issue Published : March 25, 2013

This work is licensed under a Creative Commons Attribution 4.0 International License.

Biginelli Reaction-Carboxylic Acids as Catalysts

https://doi.org/10.14233/ajchem.2013.14094

Sadia Noreen

Institute of Chemistry, University of the Punjab, Lahore, Pakistan

Saima Perveen

Department of Chemistry, The Islamia University of Bahawalpur, Bahawalpur, Pakistan

Muhammad Naeem Khan

Applied Chemistry Resarch Center, PCSIR Laboratories Complex, Lahore, Pakistan

Areesha Nazeer

Institute of Chemistry, University of the Punjab, Lahore, Pakistan

Misbahul Ain Khan

Institute of Chemistry, University of the Punjab, Lahore, Pakistan ; Department of Chemistry, The Islamia University of Bahawalpur, Bahawalpur, Pakistan

Munawar Ali Munawar

Institute of Chemistry, University of the Punjab, Lahore, Pakistan

Rabia Babar

Institute of Chemistry, University of the Punjab, Lahore, Pakistan

Farah Suhail

Institute of Chemistry, University of the Punjab, Lahore, Pakistan

Muhammad Azad

Government Polytechnic Institute for Printing and Graphic Arts, Lahore, Pakistan

Alice M.R. Bernardino

Programa de Pós- Graduação em Química, Universidade Federal Fluminense, Niterói-RJ, Brazil

Maurício S. Dos Santos

Departamento de Física e Química, Universidade Federal de Itajubá, Itajubá-MG, Brazil

Corresponding Author(s) : Muhammad Naeem Khan

changwani_1@yahoo.com

Asian Journal of Chemistry, Vol. 25 No. 9 (2013): Vol 25 Issue 9
Article Published : April 8, 2013

Abstract

Mono and dicarboxylic acids were found to be excellent catalysts for the synthesis of dihydropyrimidones/thiones. These are presented as alternate and cheap catalysts for the multicomponent reactions.

Keywords

Multicomponent reactions Dihydropyrimidone Dihydropyrimidothione Acid catalysts

Noreen, S., Perveen, S., Naeem Khan, M., Nazeer, A., Ain Khan, M., Ali Munawar, M., … S. Dos Santos, M. . (2013). Biginelli Reaction-Carboxylic Acids as Catalysts. Asian Journal of Chemistry, 25(9), 4770–4772. https://doi.org/10.14233/ajchem.2013.14094

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References

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I. Saxena, D.C. Borah and J.C. Sarma, Tetrahedron Lett., 46, 1159 (2005).
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D. Shobha, M.A. Chari, P. Sadanandam and K. Mukkanti, J. Heterocycl. Chem., 45, 1225 (2008).
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F. Tamaddon, Z. Razmi and A.A. Jafar, Tetrahedron Lett., 51, 1187 (2010).
J. Peng and Y. Deng, Tetrahedron Lett., 42, 5917 (2001).
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J. Lu and H. Ma, Synlett, 63 (2000).
Y. Yu, D. Liu, C. Liu and G. Luo, Bioorg. Med. Chem. Lett., 17, 3508 (2007).
S. Gore, S. Baskaran and B. Koenig, Green Chem., 13, 1009 (2011).
J. Wichmann, G. Adam, S. Kolczewski, V. Mutel and T. Woltering, Bioorg. Med. Chem. Lett., 9, 1573 (1999).

References

D.J. Brown, In eds.: A.R. Katritzky and C. W Rees, In Comprehensive Heterocyclic Chemistry; Pergamon Press: Oxford (1984).

P. Biginelli, Gazz. Chim. Ital., 23, 360 (1893).

G.C. Rovnyak, S.D. Kimball, B. Beyer, G. Cucinotta, J.D. Dimarco, J. Gougoutas, A. Hedberg, M. Malley, J.P. McCarthy, R. Zhang and S. Moreland, J. Med. Chem., 38, 119 (1995).

G.C. Rovnyak, K.S. Atwal, A. Hedberg, S.D. Kimball, S. Moreland, J.Z. Gougoutas, B.C. O' Reilly, J. Schwarz and M.F. Malley, J. Med. Chem., 35, 3254 (1992).

S.D. Sidler, R.D. Larsen, M. Chartrain, N. Ikemoto, C.M. Roberge, C.S. Taylor, W. Li and G.F. Bills, PCT. Int. Appl. WO# 9906795 (1999).

C.O. Kappe and A. Stadler, Org. React. A, 65, 1 (2004).

K. Ramalinga, P. Vijayalakshmi and T.N.B. Kaimal, Synlett, 863 (2001).

J. Lu and Y. Bai, Synthesis, 466 (2002).

C.V. Reddy, M. Mahesh, P.V.K. Raju, T.R. Babu and V.V.N. Reddy, Tetrahedron Lett., 43, 2657 (2002).

C. Liu, J. Wang and Y. Li, J. Mol. Catal. A, 258, 367 (2006).

L. Wang, C. Qian, H. Tian and Y. Ma, Synth. Commun., 33, 1459 (2003).

P. Salehi, M. Dabiri, M.A. Zolfigol and M.A.B. Fardi, Tetrahedron Lett., 44, 2889 (2003).

M. Kidwai, S. Saxena, R. Mohan and R. Venkataramanan, J. Chem. Soc. Perkin Trans. 1, 1845 (2002).

M. Abdollahi and Z. Zaghaghi, Chem. Papers, 63, 97 (2009).

I. Saxena, D.C. Borah and J.C. Sarma, Tetrahedron Lett., 46, 1159 (2005).

X. Feng, J.-J. Wang and Y.-P. Tian, Synth. Commun., 38, 1299 (2008).

D. Shobha, M.A. Chari, P. Sadanandam and K. Mukkanti, J. Heterocycl. Chem., 45, 1225 (2008).

D. Russowsky, F.A. Lopes, V.S.S. da Silva, K.F.S. Canto, M.G.M. D` Oca and M.N. Godoi, J. Braz. Chem. Soc., 15, 165 (2004).

A. Debache, M. Amimour, A. Belfaitah, S. Rhouati and B. Carboni, Tetrahedron Lett., 49, 6119 (2008).

F. Tamaddon, Z. Razmi and A.A. Jafar, Tetrahedron Lett., 51, 1187 (2010).

J. Peng and Y. Deng, Tetrahedron Lett., 42, 5917 (2001).

E.H. Hu, D.R. Sidler and U.H. Dolling, J. Org. Chem., 63, 3454 (1998).

J. Lu and H. Ma, Synlett, 63 (2000).

Y. Yu, D. Liu, C. Liu and G. Luo, Bioorg. Med. Chem. Lett., 17, 3508 (2007).

S. Gore, S. Baskaran and B. Koenig, Green Chem., 13, 1009 (2011).

J. Wichmann, G. Adam, S. Kolczewski, V. Mutel and T. Woltering, Bioorg. Med. Chem. Lett., 9, 1573 (1999).

Issue

Vol. 25 No. 9 (2013): Vol 25 Issue 9

Biginelli Reaction-Carboxylic Acids as Catalysts

Corresponding Author(s) : Muhammad Naeem Khan

Abstract

Keywords

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