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Vol. 22 No. 9 (2010): Vol 22 Issue 9

An Effective N-Ligand for Copper-Catalyzed N-Arylation of Triazole

Yan Yang
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China
Yong-Sheng Jin
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China
Hong-Gang Hu
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China
Qing-Jie Zhao
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China
Yan Zou
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China
Qiu-Ye Wu
Department of Organic Chemistry, School of Pharmacy, Second Military Medical University, Shanghai 200433, P.R. China

Corresponding Author(s) : Yan Yang

lululion666@163.com; wuqysmmu@sohu.com

Asian Journal of Chemistry, Vol. 22 No. 9 (2010): Vol 22 Issue 9

Abstract

An effective N-ligand for copper-catalyzed N-arylation of 1H-1,2,4-triazole has been developed. In the presence of Cu2O, Cs2CO3, N-ligand-B, 1H-1,2,4-triazole were coupled with toluene to afford the corresponding products in moderate condition and with excellent yields.

Keywords

N-Ligand C-N Bond cross-coupling Copper-catalyzed 1H-1,2,4-Triazole
(1)
Yang, Y.; Jin, Y.-S.; Hu, H.-G.; Zhao, Q.-J.; Zou, Y.; Wu, Q.-Y. An Effective N-Ligand for Copper-Catalyzed N-Arylation of Triazole. ajc 2010, 22, 7435-7437.
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